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Studi in silico di derivati ​​dell’indenopirazolo per il cancro

Studi in silico di derivati ​​dell’indenopirazolo per il cancro

Md. Muzaffar-ur- Rehman

45,16 €
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Editorial:
KS OmniScriptum Publishing
Año de edición:
2024
Materia
Química
ISBN:
9786208025083
45,16 €
IVA incluido
Disponible

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Gli indenopirazoli sono i nuovi farmaci utilizzati per curare il cancro. È stato condotto uno studio in silico per comprendere l’analogo più attivo mediante metodi 3D QSAR mediante l’implicazione di studi CoMFA e CoMSIA che ci aiuterebbero a prevedere l’attività del farmaco. Sono stati condotti anche studi di docking per determinare l’interazione degli analoghi. In questo libro è stato condotto un breve studio dell’indenopirazolo e dei suoi analoghi. Questo studio mira a progettare un modello QSAR mediante il quale può essere sviluppato un nuovo analogo che, in seguito a ulteriori studi, potrebbe agire come un potente inibitore di cdk4 per curare il cancro.

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